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For research and educational purposes only. Not intended for human consumption.

Melanotan II

Well Researched
Updated Dec 2025

Synthetic Melanocortin Peptide | Tanning & Sexual Function

InjectableTopicalNasal
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0.25-1mg
1-2x daily
Injectable
Subcutaneous: abdomen (preferred)
4-8 weeks
Typical duration
2-8°C
Refrigerated

Overview

What is Melanotan II?

Melanotan II is a synthetic analog of alpha-melanocyte-stimulating hormone (α-MSH) that stimulates melanin production for skin tanning and has additional effects on sexual arousal and appetite suppression. Originally developed at the University of Arizona as a sunless tanning agent, it has gained attention for its dual effects on pigmentation and sexual function through melanocortin receptor activation.

Key Benefits

Rapid tanning without UV exposure, enhanced libido and sexual function, appetite suppression, and improved mood through melanocortin activation.

Mechanism of Action

Binds to melanocortin receptors (MC1R, MC3R, MC4R, MC5R) throughout the body. MC1R activation stimulates melanocytes to produce eumelanin, while MC4R affects sexual arousal and appetite regulation.

Molecular Information

1,024.18 Da
Weight
7
amino acids
Melanocortin receptor agonist
Type
Amino Acid Sequence:
Ac-Nle-cyclo[Asp-His-D-Phe-Arg-Trp-Lys]-NH₂
* Cyclic peptide structure for enhanced receptor binding and stability

Pharmacokinetics

Peak
30 min
Half-life
1 hr
Cleared
~5 hrs
100%50%0%0h6h12h18h24h
Peak
Half-life
Cleared
Dorr et al. 1996

Research Indications

UV-Free Tanning

Stimulates natural melanin production for darker skin tone without sun damage.

Photoprotection

Increased melanin provides natural SPF and reduces sunburn risk.

Even Pigmentation

Promotes uniform tanning and may help with certain pigmentation disorders.

Research Protocols

Disclaimer: Melanotan II is not approved for human use. These are commonly discussed research protocols. Consult a healthcare provider before use.

GoalDoseFrequencyRoute
Initial Loading0.25mgDailySubcutaneous
Tanning Maintenance0.5-1mg2-3x weeklySubcutaneous
Sexual Enhancement0.5-1mgAs neededSubcutaneous
Minimal Side Effects0.1-0.25mgEvery other daySubcutaneous
Photoprotection0.5mg2x weeklySubcutaneous

Timing: For tanning: morning dosing preferred. For sexual effects: 2-4 hours before activity. Can split daily dose to minimize side effects.

Peptide Interactions

How to Reconstitute

Important: Always use bacteriostatic water (BAC). Sterile technique is essential.

1

Clean vial tops with alcohol swab and let dry

2

Draw 2ml bacteriostatic water for 10mg vial (creates 5mg/ml concentration)

3

Inject water slowly down the side of peptide vial to avoid foaming

4

Gently roll vial between hands - do not shake vigorously

5

Solution should be clear to slightly yellow

6

Store reconstituted peptide in refrigerator wrapped in foil (light sensitive)

7

Draw dose with insulin syringe - typical dose is 0.05-0.2ml

Dosing Calculator

Calculate your injection volume with visual dosing guide

FINAL CONCENTRATION
2.50mg/mL
Each milliliter contains 2.50 mg of peptide
VISUAL REFERENCE (RESEARCH USE ONLY)

To obtain 250 mcg from this solution:

Draw 0.10 mL=10 units

(1 mL = 100 units on any insulin syringe)

0102030405060708090100
00.10.20.30.40.50.60.70.80.91.0
0.10 mL
10 units

Draw to this mark for 250 mcg

This calculator is for research purposes only. Always verify calculations and consult protocols.

Quality Indicators

White to Off-White Lyophilized Powder

Pure MT-II appears as white or slightly off-white powder before reconstitution.

Clear to Pale Yellow When Reconstituted

Properly mixed solution should be transparent with at most a slight yellow tint.

Protect From Light Exposure

MT-II is photosensitive - wrap vial in foil and minimize light exposure.

Brown or Dark Colored Powder

Indicates oxidation or impurities - do not use.

Cloudy Solution After Mixing

Suggests degradation or contamination - discard immediately.

What to Expect

  • Day 1-3: Possible nausea, flushing, and fatigue after injection
  • Day 3-7: Increased spontaneous erections (men), enhanced arousal
  • Week 1-2: Noticeable skin darkening, reduced appetite
  • Week 2-4: Significant tanning, stabilized sexual effects
  • Week 4+: Maintained tan with less frequent dosing

Side Effects & Safety

Side Effects

  • Start with very low dose (0.1-0.25mg) to assess tolerance
  • Nausea is common - can pre-treat with antiemetic if needed
  • Monitor moles and freckles for changes in size or color
  • Stay hydrated to minimize headaches and flushing
  • Avoid if history of melanoma or dysplastic nevi
  • Blood pressure may increase temporarily after injection

When to Stop

  • New or changing moles
  • Severe nausea or vomiting
  • Significant blood pressure changes
  • Allergic reactions
  • Facial flushing that doesn't resolve
  • Consult dermatologist for any skin concerns

References

3 Studies

Photoprotection in Fair-Skinned Individuals

Human (Fitzpatrick Type I-II) | 0.1mg/kg | 3 months | Reduced sunburn incidence

Long-term study showed sustained increase in melanin production and significant reduction in UV-induced erythema in individuals with high sunburn susceptibility.

Female Sexual Arousal Disorder Trial

Human (Female) | 0.025mg/kg | Single dose | 73% reported arousal

Crossover study in premenopausal women with sexual arousal disorder showed significant increases in genital arousal and sexual desire within 24 hours.

Cardiovascular Effects Assessment

Human | Various doses | Acute monitoring | Mild BP elevation

Comprehensive cardiovascular monitoring revealed transient increases in blood pressure and heart rate, typically mild and self-limiting.

Quick Start Guide

Typical Dose
0.25-1mg
How Often
Daily initially, then 2-3x weekly for maintenance
Where to Inject
Subcutaneous: abdomen (preferred)
Timing
Morning for tanning, 2-4 hours before activity for sexual effects
Effects Timeline
Tanning: 7-10 days, Sexual: 2-4 hours, Appetite: immediate
Storage
Refrigerate, protect from light
Cycle Length
4-8 weeks on, 4 weeks off
Break Between
4 weeks minimum to assess melanin fading

Research Disclaimer

Melanotan II is sold for laboratory research purposes only and is not intended for human or animal consumption. The information provided on this page is compiled from published research, veterinary studies, and anecdotal reports for educational purposes. This content does not constitute medical advice, diagnosis, or treatment recommendations. Any research involving Melanotan II must comply with all applicable local, state, and federal regulations. BioInfinity Lab makes no claims regarding the safety or efficacy of Melanotan II for any purpose. Consult qualified professionals for any research applications.